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Smedley, C. J., Li, G., Barrow, A. S., Gialelis, T. L., Giel, M. C., Ottonello, A., Cheng, Y., Kitamura, S., Wolan, D. W., Sharpless, K. B., Moses, J. E. (April 2020) Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores from 2-Substituted-Alkynyl-1-Sulfonyl Fluoride (SASF) Hubs. Angew Chem Int Ed Engl. ISSN 1433-7851
Giel, M. C., Smedley, C. J., Mackie, E. R. R., Guo, T., Dong, J., Soares da Costa, T. P., Moses, J. E. (January 2020) Metal-Free Synthesis of Functional 1-Substituted-1,2,3-Triazoles from Ethenesulfonyl Fluoride and Organic Azides. Angew Chem Int Ed Engl, 59 (3). pp. 1181-1186. ISSN 1433-7851
Suhua, Li, Gencheng, Li, Bing, Gao, Sidharam P., Pujari, Xiaoyan, Chen, Hyunseok, Kim, Feng, Zhou, Liana M., Klivansky, Yi, Liu, Hafedh, Driss, Rachael E., Impey, Tatiana P. Soares da, Costa, Jianmei, Lu, Peng, Wu, Han, Zuilhof, John E., Moses, K. Barry, Sharpless (October 2019) SuFExable Polymers with Helical Structures Derived from Thionyl Tetrafluoride (SOF4). chemRxiv. (Unpublished)
Zheng, Q., Woehl, J. L., Kitamura, S., Santos-Martins, D., Smedley, C. J., Li, G., Forli, S., Moses, J. E., Wolan, D. W., Sharpless, K. B. (September 2019) SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase. Proc Natl Acad Sci U S A, 116 (38). pp. 18808-18814. ISSN 0027-8424 (Print)0027-8424
Barrow, A. S., Smedley, C. J., Zheng, Q., Li, S., Dong, J., Moses, J. E. (August 2019) The growing applications of SuFEx click chemistry. Chem Soc Rev, 48 (17). pp. 4731-4758. ISSN 0306-0012
Liu, F., Wang, H., Li, S., Bare, G. A. L., Chen, X., Wang, C., Moses, J. E., Wu, P., Sharpless, K. B. (June 2019) Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF(4) )-Derived Connective Hubs for Bioconjugation to DNA and Proteins. Angew Chem Int Ed Engl, 58 (24). pp. 8029-8033. ISSN 1433-7851 (Print)1433-7851
Smedley, C. J., Zheng, Q., Gao, B., Li, S., Molino, A., Duivenvoorden, H. M., Parker, B. S., Wilson, D. J. D., Sharpless, K. B., Moses, J. E. (March 2019) Bifluoride Ion Mediated SuFEx Trifluoromethylation of Sulfonyl Fluorides and Iminosulfur Oxydifluorides. Angew Chem Int Ed Engl, 58 (14). pp. 4552-4556. ISSN 1433-7851
Randall, J. D., Eyckens, D. J., Stojcevski, F., Francis, P. S., Doeven, E. H., Barlow, A. J., Barrow, A. S., Arnold, C. L., Moses, J. E., Henderson, L. C. (September 2018) Modification of Carbon Fibre Surfaces by Sulfur-Fluoride Exchange Click Chemistry. Chemphyschem. ISSN 1439-4235
Gahtory, D., Sen, R., Pujari, S., Li, S., Zheng, Q., Moses, J. E., Sharpless, K. B., Zuilhof, H. (July 2018) Quantitative and Orthogonal Formation and Reactivity of SuFEx Platforms. Chemistry, 24 (41). pp. 10550-10556. ISSN 0947-6539 (Print)0947-6539
Sharma, P., Bhat, S. V., Prabhath, M. R. R., Molino, A., Nauha, E., Wilson, D. J. D., Moses, J. E. (July 2018) Synthesis of 1,2,4-Triazol-3-imines via Selective Stepwise Cycloaddition of Nitrile Imines with Organo-cyanamides. Org Lett, 20 (14). pp. 4263-4266. ISSN 1523-7052
Smedley, C. J., Stanley, P. A., Qazzaz, M. E., Prota, A. E., Olieric, N., Collins, H., Eastman, H., Barrow, A. S., Lim, K. H., Kam, T. S., Smith, B. J., Duivenvoorden, H. M., Parker, B. S., Bradshaw, T. D., Steinmetz, M. O., Moses, J. E. (July 2018) Sustainable Syntheses of (-)-Jerantinines A & E and Structural Characterisation of the Jerantinine-Tubulin Complex at the Colchicine Binding Site. Sci Rep, 8 (1). p. 10617. ISSN 2045-2322
Smedley, C. J., Giel, M. C., Molino, A., Barrow, A. S., Wilson, D. J. D., Moses, J. E. (June 2018) 1-Bromoethene-1-sulfonyl fluoride (BESF) is another good connective hub for SuFEx click chemistry. Chem Commun (Camb), 54 (47). pp. 6020-6023. ISSN 1359-7345
Powell, Kimberley J., Richens, Joanna L., Bramble, Jonathan P., Han, Li-Chen, Sharma, Pallavi, O'Shea, Paul, Moses, John E. (March 2018) Photochemical activity of membrane-localised polyketide derived marine natural products. Tetrahedron, 74 (12). pp. 1191-1198. ISSN 0040-4020
Jenner, M., Kosol, S., Griffiths, D., Prasongpholchai, P., Manzi, L., Barrow, A. S., Moses, J. E., Oldham, N. J., Lewandowski, J. R., Challis, G. L. (March 2018) Mechanism of intersubunit ketosynthase-dehydratase interaction in polyketide synthases. Nat Chem Biol, 14 (3). pp. 270-275. ISSN 1552-4450 (Print)1552-4450
Gao, B., Li, S., Wu, P., Moses, J. E., Sharpless, K. B. (February 2018) SuFEx Chemistry of Thionyl Tetrafluoride (SOF(4) ) with Organolithium Nucleophiles: Synthesis of Sulfonimidoyl Fluorides, Sulfoximines, Sulfonimidamides, and Sulfonimidates. Angew Chem Int Ed Engl, 57 (7). pp. 1939-1943. ISSN 1433-7851 (Print)1433-7851
Manzi, L., Barrow, A. S., Hopper, J. T. S., Kaminska, R., Kleanthous, C., Robinson, C. V., Moses, J. E., Oldham, N. J. (November 2017) Carbene Footprinting Reveals Binding Interfaces of a Multimeric Membrane-Spanning Protein. Angew Chem Int Ed Engl, 56 (47). pp. 14873-14877. ISSN 1433-7851
Smedley, C. J., Barrow, A. S., Spiteri, C., Giel, M. C., Sharma, P., Moses, J. E. (July 2017) Sulfur-Fluoride Exchange (SuFEx)-Mediated Synthesis of Sterically Hindered and Electron-Deficient Secondary and Tertiary Amides via Acyl Fluoride Intermediates. Chemistry, 23 (42). pp. 9990-9995. ISSN 0947-6539
Li, S., Wu, P., Moses, J. E., Sharpless, K. B. (March 2017) Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF(4) Hub. Angew Chem Int Ed Engl, 56 (11). pp. 2903-2908. ISSN 1433-7851 (Print)1433-7851
Silverman, S. M., Moses, J. E., Sharpless, K. B. (January 2017) Reengineering Antibiotics to Combat Bacterial Resistance: Click Chemistry [1,2,3]-Triazole Vancomycin Dimers with Potent Activity against MRSA and VRE. Chemistry, 23 (1). pp. 79-83. ISSN 0947-6539
Manzi, L., Barrow, A. S., Scott, D., Layfield, R., Wright, T. G., Moses, J. E., Oldham, N. J. (November 2016) Carbene footprinting accurately maps binding sites in protein-ligand and protein-protein interactions. Nat Commun, 7. p. 13288. ISSN 2041-1723
Han, L. C., Stanley, P. A., Wood, P. J., Sharma, P., Kuruppu, A. I., Bradshaw, T. D., Moses, J. E. (August 2016) Horner-Wadsworth-Emmons approach to piperlongumine analogues with potent anti-cancer activity. Org Biomol Chem, 14 (31). pp. 7585-93. ISSN 1477-0520
Barrow, A. S., Moses, J. E. (July 2016) Synthesis of Sulfonyl Azides via Lewis Base Activation of Sulfonyl Fluorides and Trimethylsilyl Azide. Synlett, 27 (12). pp. 1840-1843. ISSN 0936-5214
Zhang, E., Tang, J., Li, S., Wu, P., Moses, J. E., Sharpless, K. B. (April 2016) Chemoselective Synthesis of Polysubstituted Pyridines from Heteroaryl Fluorosulfates. Chemistry, 22 (16). pp. 5692-7. ISSN 0947-6539 (Print)0947-6539
Bhat, S. V., Robinson, D., Moses, J. E., Sharma, P. (March 2016) Synthesis of Oxadiazol-5-imines via the Cyclizative Capture of in Situ Generated Cyanamide Ions and Nitrile Oxides. Org Lett, 18 (5). pp. 1100-3. ISSN 1523-7052
Stanley, P. A., Spiteri, C., Moore, J. C., Barrow, A. S., Sharma, P., Moses, J. E. (January 2016) Biomimetic Approaches Towards The Synthesis of Complex Dimeric Natural Products. Curr Pharm Des, 22 (12). pp. 1628-57. ISSN 1381-6128
Roe, S., Gunaratnam, M., Spiteri, C., Sharma, P., Alharthy, R. D., Neidle, S., Moses, J. E. (August 2015) Synthesis and biological evaluation of hybrid acridine-HSP90 ligand conjugates as telomerase inhibitors. Org Biomol Chem, 13 (31). pp. 8500-4. ISSN 1477-0520
Cousins, A. R., Ritson, D., Sharma, P., Stevens, M. F., Moses, J. E., Searle, M. S. (December 2014) Ligand selectivity in stabilising tandem parallel folded G-quadruplex motifs in human telomeric DNA sequences. Chem Commun (Camb), 50 (96). pp. 15202-5. ISSN 1359-7345
Moore, J. C., Davies, E. S., Walsh, D. A., Sharma, P., Moses, J. E. (October 2014) Formal synthesis of kingianin A based upon a novel electrochemically-induced radical cation Diels-Alder reaction. Chem Commun (Camb), 50 (83). pp. 12523-5. ISSN 1359-7345
Dempster, S., Harper, S., Moses, J. E., Dreveny, I. (May 2014) Structural characterization of the apo form and NADH binary complex of human lactate dehydrogenase. Acta Crystallogr D Biol Crystallogr, 70 (Pt 5). pp. 1484-90. ISSN 0907-4449 (Print)0907-4449
Powell, K. J., Han, L. C., Sharma, P., Moses, J. E. (April 2014) Chemoselective palladium-catalyzed cyanation of alkenyl halides. Org Lett, 16 (8). pp. 2158-61. ISSN 1523-7052
Carbone, G., Burnley, J., Moses, J. E. (April 2013) A catalytic and tert-butoxide ion-mediated amidation of aldehydes with para-nitro azides. Chem Commun (Camb), 49 (27). pp. 2759-61. ISSN 1359-7345
Sharma, P., Ritson, D. J., Burnley, J., Moses, J. E. (October 2011) A synthetic approach to kingianin A based on biosynthetic speculation. Chem Commun (Camb), 47 (38). pp. 10605-7. ISSN 1359-7345
Ritson, D. J., Spiteri, C., Moses, J. E. (May 2011) A silver-mediated one-step synthesis of oxazoles. J Org Chem, 76 (9). pp. 3519-22. ISSN 0022-3263
Moorhouse, A. D., Spiteri, C., Sharma, P., Zloh, M., Moses, J. E. (January 2011) Targeting glycolysis: a fragment based approach towards bifunctional inhibitors of hLDH-5. Chem Commun (Camb), 47 (1). pp. 230-2. ISSN 1359-7345
Spiteri, C., Keeling, S., Moses, J. E. (August 2010) New synthesis of 1-substituted-1H-indazoles via 1,3-dipolar cycloaddition of in situ generated nitrile imines and benzyne. Org Lett, 12 (15). pp. 3368-71. ISSN 1523-7052
Roe, S., Ritson, D. J., Garner, T., Searle, M., Moses, J. E. (June 2010) Tuneable DNA-based asymmetric catalysis using a G-quadruplex supramolecular assembly. Chem Commun (Camb), 46 (24). pp. 4309-11. ISSN 1359-7345
Sharma, P., Moses, J. E. (June 2010) Ethynyldiisopropylsilyl: a new alkynylsilane protecting group and "click" linker. Org Lett, 12 (12). pp. 2860-3. ISSN 1523-7052
Spiteri, C., Mason, C., Zhang, F., Ritson, D. J., Sharma, P., Keeling, S., Moses, J. E. (June 2010) An efficient entry to 1,2-benzisoxazoles via 1,3-dipolar cycloaddition of in situ generated nitrile oxides and benzyne. Org Biomol Chem, 8 (11). pp. 2537-42. ISSN 1477-0520
Sharma, P., Moses, J. E. (March 2010) Photochemical Studies of the Tridachiahydropyrones in Seawater. Synlett (4). pp. 525-528. ISSN 0936-5214
Spiteri, C., Sharma, P., Zhang, F., Macdonald, S. J., Keeling, S., Moses, J. E. (February 2010) An improved synthesis of 1,2-benzisoxazoles: TBAF mediated 1,3-dipolar cycloaddition of nitrile oxides and benzyne. Chem Commun (Camb), 46 (8). pp. 1272-4. ISSN 1359-7345
Spiteri, C., Moses, J. E. (January 2010) Copper-catalyzed azide-alkyne cycloaddition: regioselective synthesis of 1,4,5-trisubstituted 1,2,3-triazoles. Angew Chem Int Ed Engl, 49 (1). pp. 31-3. ISSN 1433-7851
Garner, T. P., Williams, H. E., Gluszyk, K. I., Roe, S., Oldham, N. J., Stevens, M. F., Moses, J. E., Searle, M. S. (October 2009) Selectivity of small molecule ligands for parallel and anti-parallel DNA G-quadruplex structures. Org Biomol Chem, 7 (20). pp. 4194-200. ISSN 1477-0520
Moses, John E., Rueping, Magnus, Cronin, Leroy (September 2009) Highlights from the 44th EUCHEM Conference on Stereochemistry, Bürgenstock, Switzerland, May 2009. Chemical Communications (41). pp. 6125-6128. ISSN 1359-7345
Gunaratnam, M., Green, C., Moreira, J. B., Moorhouse, A. D., Kelland, L. R., Moses, J. E., Neidle, S. (July 2009) G-quadruplex compounds and cis-platin act synergistically to inhibit cancer cell growth in vitro and in vivo. Biochem Pharmacol, 78 (2). pp. 115-22. ISSN 0006-2952
Sharma, P., Lygo, B., Lewis, W., Moses, J. E. (April 2009) Biomimetic synthesis and structural reassignment of the tridachiahydropyrones. J Am Chem Soc, 131 (16). pp. 5966-72. ISSN 0002-7863
Zhang, F., Moses, J. E. (April 2009) Benzyne click chemistry with in situ generated aromatic azides. Org Lett, 11 (7). pp. 1587-90. ISSN 1523-7052
Sharma, P., Griffiths, N., Moses, J. E. (September 2008) Biomimetic synthesis and structural revision of (+/-)-tridachiahydropyrone. Org Lett, 10 (18). pp. 4025-7. ISSN 1523-7052
Moorhouse, A. D., Moses, J. E. (August 2008) Microwave enhancement of a 'one-pot' tandem azidation-'click' cycloaddition of anilines. Synlett (14). pp. 2089-2092. ISSN 0936-5214
Eade, S. J., Walter, M. W., Byrne, C., Odell, B., Rodriguez, R., Baldwin, J. E., Adlington, R. M., Moses, J. E. (July 2008) Biomimetic synthesis of pyrone-derived natural products: exploring chemical pathways from a unique polyketide precursor. J Org Chem, 73 (13). pp. 4830-9. ISSN 0022-3263
Moorhouse, A. D., Haider, S., Gunaratnam, M., Munnur, D., Neidle, S., Moses, J. E. (June 2008) Targeting telomerase and telomeres: a click chemistry approach towards highly selective G-quadruplex ligands. Mol Biosyst, 4 (6). pp. 629-42. ISSN 1742-2051
Moorhouse, A. D., Moses, J. E. (May 2008) Click chemistry and medicinal chemistry: a case of "cyclo-addiction". ChemMedChem, 3 (5). pp. 715-23. ISSN 1860-7179
Moses, J. E., Moorhouse, A. D. (August 2007) The growing applications of click chemistry. Chemical Society Reviews, 36 (8). pp. 1249-1262. ISSN 0306-0012
Rodriguez, R., Adlington, R. M., Eade, S. J., Walter, M. W., Baldwin, J. E., Moses, J. E. (May 2007) Total synthesis of cyercene A and the biomimetic synthesis of (+/-)-9,10-deoxytridachione and (+/-)-ocellapyrone A. Tetrahedron, 63 (21). pp. 4500-4509. ISSN 0040-4020
Barral, K., Moorhouse, A. D., Moses, J. E. (April 2007) Efficient conversion of aromatic amines into azides: a one-pot synthesis of triazole linkages. Org Lett, 9 (9). pp. 1809-11. ISSN 1523-7060 (Print)1523-7052
Moorhouse, A. D., Santos, A. M., Gunaratnam, M., Moore, M., Neidle, S., Moses, J. E. (December 2006) Stabilization of G-quadruplex DNA by highly selective ligands via click chemistry. J Am Chem Soc, 128 (50). pp. 15972-3. ISSN 0002-7863 (Print)0002-7863
Comméiras, Laurent, Moses, John E., Adlington, Robert M., Baldwin, Jack E., Cowley, Andrew R., Baker, Christopher M., Albrecht, Birgit, Grant, Guy H. (October 2006) Total synthesis of the epoxyquinol dimer (+)-panepophenanthrin: application of a diastereospecific biomimetic Diels–Alder dimerisation. Tetrahedron, 62 (42). pp. 9892-9901. ISSN 0040-4020
Jacobsen, Mikkel F., Moses, John E., Adlington, Robert M., Baldwin, Jack E. (2006) The biomimetic synthesis of SNF4435C and SNF4435D, and the total synthesis of the polyene metabolites aureothin, N-acetyl-aureothamine and spectinabilin. Tetrahedron, 62 (8). pp. 1675-1689. ISSN 0040-4020
Moses, J. E., Adlington, R. M. (December 2005) Sir Jack Baldwin, FRS: biomimetic studies at Oxford. Chem Commun (Camb), 48. pp. 5945-52. ISSN 1359-7345 (Print) 1359-7345
Rodriguez, R., Moses, J. E., Adlington, R. M., Baldwin, J. E. (October 2005) A new and efficient method for o-quinone methide intermediate generation: application to the biomimetic synthesis of the benzopyran derived natural products (+/-)-lucidene and (+/-)-alboatrin. Org Biomol Chem, 3 (19). pp. 3488-95. ISSN 1477-0520 (Print)1477-0520
Jacobsen, M. F., Moses, J. E., Adlington, R. M., Baldwin, J. E. (June 2005) The total synthesis of spectinabilin and its biomimetic conversion to SNF4435C and SNF4435D. Org Lett, 7 (12). pp. 2473-6. ISSN 1523-7060 (Print)1523-7052
Moses, J. E., Adlington, R. M., Rodriguez, R., Eade, S. J., Baldwin, J. E. (April 2005) Biomimetic synthesis of (+/-)-9,10-deoxytridachione. Chem Commun (Camb) (13). pp. 1687-9. ISSN 1359-7345 (Print)1359-7345
Rodriguez, R., Adlington, R. M., Moses, J. E., Cowley, A., Baldwin, J. E. (September 2004) A new and efficient method for o-quinone methide intermediate generation: application to the biomimetic synthesis of (+/-)-Alboatrin. Org Lett, 6 (20). pp. 3617-9. ISSN 1523-7060 (Print)1523-7052
Moses, John E., Baldwin, Jack E., Adlington, Robert M. (August 2004) An efficient synthesis of cyercene A. Tetrahedron Letters, 45 (34). pp. 6447-6448. ISSN 0040-4039
Moses, J. E., Baldwin, J. E., Brückner, S., Eade, S. J., Adlington, R. M. (November 2003) Biomimetic studies on polyenes. Org Biomol Chem, 1 (21). pp. 3670-84. ISSN 1477-0520 (Print) 1477-0520
Moses, John E., Baldwin, Jack E., Adlington, Robert M., Cowley, Andrew R., Marquez, Rodolfo (August 2003) Thermally induced cascade pericyclic reaction pathways from tetraene esters. Tetrahedron Letters, 44 (35). pp. 6625-6627. ISSN 0040-4039
Moses, J. E., Commeiras, L., Baldwin, J. E., Adlington, R. M. (August 2003) Total synthesis of panepophenanthrin. Org Lett, 5 (17). pp. 2987-8. ISSN 1523-7060 (Print)1523-7052
Son, A. J. R., Schweiger, S. W., Thorn, M. G., Moses, J. E., Fanwick, P. E., Rothwell, I. P. (April 2003) The isolation and chemistry of tantalum dimethylamides containing resolved 3,3 '-disubstituted-1,1 '-bi-2,2 '-naphthoxide ligands. Dalton Transactions (8). pp. 1620-1627. ISSN 1477-9226
Moses, J. E., Baldwin, J. E., Marquez, R., Adlington, R. M., Claridge, T. D., Odell, B. (March 2003) Biomimetic synthesis of the crispatene core. Org Lett, 5 (5). pp. 661-3. ISSN 1523-7060 (Print)1523-7052
Moses, J. E., Baldwin, J. E., Marquez, R., Adlington, R. M., Cowley, A. R. (October 2002) Studies on the biomimetic synthesis of SNF4435 C and D. Org Lett, 4 (21). pp. 3731-4. ISSN 1523-7060 (Print)1523-7052
Thorn, M. G., Moses, J. E., Fanwick, P. E., Rothwell, I. P. (January 2000) New tantalum compounds supported by 3,3 '-disubstituted-1,1 '-bi-2-naphthoxide ligation. Journal of the Chemical Society-Dalton Transactions (16). pp. 2659-2660. ISSN 1470-479X
Burnley, J., Ralph, M., Sharma, P., Moses, J. E. (2011) Biomimetic Electrocyclization Reactions toward Polyketide-Derived Natural Products. In: Biomimetic Organic Synthesis. John Wiley & Sons, pp. 591-635. ISBN 9783527634606
Abdullah, Nurul Akmaryanti, Moses, John, Han, Li Chen, Storr, Sarah, Ammar, Aula, Martin, Stewart G. (July 2017) Abstract 5210: Differential cytotoxic effects of Piperlongumine analogues and their radiotherapeutic response in breast cancer. In: UNSPECIFIED.
Qinheng, Zheng, Jordan L., Woehl, Seiya, Kitamura, Diogo, Santos-Martins, Christopher J., Smedley, Gencheng, Li, Stefano, Forli, John E., Moses, Dennis W., Wolan, K. Barry, Sharpless (March 2019) "Sleeping Beauty" Phenomenon: SuFEx-Enabled Discovery of Selective Covalent Inhibitors of Human Neutrophil Elastase. UNSPECIFIED. (Unpublished)
